· Introduction: mannitol
· Cerebral
· Circulatory
· Renal
Summary |
· Large (182g/mol) and polar hence does not cross cell membranes including blood-brain barrier · Substance derived from mannose, a monosaccharide · Uses: emergency reduction in ICP, osmotic diuresis |
Numbers |
· 20% mannitol -> 200mg/mL –> 1100mOsmol/L (cf. plasma 290mOsmol/L) · 20% 500mL = 550mosmoles |
Phases |
· Volume expansion (VE): ↑500mL plasma volume, ↑plasma osmolality -> contraction of ICF · Volume contraction (VC): osmotic diuresis, ↓plasma volume |
VE |
Direct: · Mannitol freely filtered, not reabsorbed, not secreted · ↑Tonicity of glomerular filtrate -> impairment of proximal tubular reabsorption (most important effect) · ↑Renal plasma flow rate, washout of medullary interstitium · ↑Urine flow rate (osmotic drag) · Does not protect against renal failure Compensation: · ↑ Na+/K+ exchange in distal nephron -> ↑Na+, ↓K+ (due to high flow rate) |
VC |
Direct: · ↓GFR if mAP <70 Compensation: · ↑ Na+/K+ exchange in distal nephron -> ↑Na+, ↓K+ (due to aldosterone) |
VE |
Direct: · ↑Preload -> risk of APO · ↓Viscosity -> ↑regional microcirculatory flow (incl. CNS) · Thrombophlebitis (hence require CVC) Compensation: · ANP: ↑RA stretch -> ↑release -> diuresis, natriuresis |
VC |
Direct: · ↓Preload -> ↓CO, ↓mAP, ↓cerebral perfusion · ↑Viscosity -> ↓regional microcirculatory flow · Vascular irritation Compensation: · RAAS: ↓mAP -> ↑renin/angiotensin 2/aldosterone -> ↑Na+ and H2O reabsorption, vasoconstriction · ADH: ↓blood volume (if 10%) -> ↑release -> ↑H2O reabsorption · SNS: ↓blood vol -> ↑release -> vasoconstriction, ↑CO |
VE |
· Osmotic dehydration -> ↓CNS volume -↓ICP · Only occurs if BBB intact · Peak effect 30-45mins, duration 6 hours |
VC |
· Production of idiogenic osmoles (glycine, glutamine, taurine, inositol etc.) · Hence risk of rebound cerebral oedema |
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